1017682-66-4
1017682-66-4 structure
- Name: PK 44 phosphate
- Chemical Name: PK 44 phosphate
- CAS Number: 1017682-66-4
- Molecular Formula: C17H16F5N7O•H3PO4
- Molecular Weight: 527.34
- Catalog: Signaling Pathways Metabolic Enzyme/Protease Dipeptidyl Peptidase
- Create Date: 2022-03-28 18:48:55
- Modify Date: 2024-01-12 23:37:48
-
PK44 phosphate is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 value of 15.8 nM[1].
| Name | PK 44 phosphate |
|---|---|
| Synonyms |
(3R)-3-Amino-4-(6,7-difluoro-1H-indazol-3-yl)-1-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl]-1-butanone phosphate (1:1)
(3R)-3-Amino-4-(6,7-difluoro-1H-indazol-3-yl)-1-[5,6-dihydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazin-7(8H)-yl]-1-butanone phosphate 1-Butanone, 3-amino-4-(6,7-difluoro-1H-indazol-3-yl)-1-[5,6-dihydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazin-7(8H)-yl]-, (3R)-, phosphate (1:1) |
| Description | PK44 phosphate is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 value of 15.8 nM[1]. |
|---|---|
| Related Catalog | |
| Target |
IC50: 15.8 nM (DPP-IV)[1] |
| References |
[1]. Adrian Maddaford, et al. Indazoles for use as dpp-iv inhibitors. WO2008040995A1 (compound 67) |
| Molecular Formula | C17H16F5N7O•H3PO4 |
|---|---|
| Molecular Weight | 527.34 |
| Exact Mass | 527.110535 |