PK 44 phosphate

Modify Date: 2024-01-12 23:37:48

PK 44 phosphate Structure
PK 44 phosphate structure
Common Name PK 44 phosphate
CAS Number 1017682-66-4 Molecular Weight 527.34
Density N/A Boiling Point N/A
Molecular Formula C17H16F5N7O•H3PO4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of PK 44 phosphate


PK44 phosphate is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 value of 15.8 nM[1].

 Names

Name PK 44 phosphate
Synonym More Synonyms

 PK 44 phosphate Biological Activity

Description PK44 phosphate is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 value of 15.8 nM[1].
Related Catalog
Target

IC50: 15.8 nM (DPP-IV)[1]

References

[1]. Adrian Maddaford, et al. Indazoles for use as dpp-iv inhibitors. WO2008040995A1 (compound 67)

 Chemical & Physical Properties

Molecular Formula C17H16F5N7O•H3PO4
Molecular Weight 527.34
Exact Mass 527.110535

 Synonyms

(3R)-3-Amino-4-(6,7-difluoro-1H-indazol-3-yl)-1-[3-(trifluoromethyl)-5,6-dihydro[1,2,4]triazolo[4,3-a]pyrazin-7(8H)-yl]-1-butanone phosphate (1:1)
(3R)-3-Amino-4-(6,7-difluoro-1H-indazol-3-yl)-1-[5,6-dihydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazin-7(8H)-yl]-1-butanone phosphate
1-Butanone, 3-amino-4-(6,7-difluoro-1H-indazol-3-yl)-1-[5,6-dihydro-3-(trifluoromethyl)-1,2,4-triazolo[4,3-a]pyrazin-7(8H)-yl]-, (3R)-, phosphate (1:1)