Name | JG26 |
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Description | JG26 is an ADAM17 inhibitor, with IC50 values of 12 nM, 1.9 nM, 150 nM and 9.4 nM for ADAM8, ADAM17, ADAM10 and MMP-12, respectively[1]. |
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Related Catalog | |
Target |
ADAM17:1.9 nM (IC50) ADAM8:12 nM (IC50) ADAM10:150 nM (IC50) MMP-9:>500000 nM (IC50) MMP-8:240 nM (IC50) MMP-9:1630 nM (IC50) MMP-12:9.4 nM (IC50) MMP14:19500 nM (IC50) |
References |
Molecular Formula | C19H22Br2N4O6S |
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Molecular Weight | 594.27 |