2402735-14-0

2402735-14-0 structure

Name: DPP-4 inhibitor 3
Chemical Name: DPP-4 inhibitor 3
CAS Number: 2402735-14-0
Molecular Formula: C₁₉H₂₂N₆O₂
Molecular Weight: 366.42
Catalog: Signaling Pathways Metabolic Enzyme/Protease Dipeptidyl Peptidase
Create Date: 2022-06-26 14:15:39
Modify Date: 2024-01-18 07:27:52
DPP-4 inhibitor 3 (Compound 5a) is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 of 0.75 nM. DPP-4 inhibitor 3 shows excellent antioxidant and insulinotropic activity[1].

Name	DPP-4 inhibitor 3

Description	DPP-4 inhibitor 3 (Compound 5a) is a potent dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 of 0.75 nM. DPP-4 inhibitor 3 shows excellent antioxidant and insulinotropic activity[1].
Related Catalog	Signaling Pathways >> Metabolic Enzyme/Protease >> Dipeptidyl Peptidase Signaling Pathways >> Protein Tyrosine Kinase/RTK >> ROS Research Areas >> Metabolic Disease
Target	IC50: 0.75 nM (DPP-IV)[1]
References	[1]. Bindu B, et al. Synthesis and discovery of triazolo-pyridazine-6-yl-substituted piperazines as effective anti-diabetic drugs; evaluated over dipeptidyl peptidase-4 inhibition mechanism and insulinotropic activities. Eur J Med Chem. 2020 Feb 1;187:111912.

Molecular Formula	C₁₉H₂₂N₆O₂
Molecular Weight	366.42