GSK 1562590 hydrochloride
Modify Date: 2025-08-25 18:54:44
GSK 1562590 hydrochloride structure
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Common Name | GSK 1562590 hydrochloride | ||
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| CAS Number | 1003878-07-6 | Molecular Weight | 617.95 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C30H31Cl3N4O4 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of GSK 1562590 hydrochlorideGSK 1562590 hydrochloride is a high affinity and selective antagonist of urotensin-II receptor (UT), with pKis of 9.14-9.66 for mammalian recombinant (mouse, rat, cat, monkey, human) and native UT[1]. |
| Name | 4'-[(1R)-1-{[(6,7-Dichloro-3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)acetyl](methyl)amino}-2-(1-pyrrolidinyl)ethyl]-3-biphenylcarboxamide hydrochloride (1:1) |
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| Synonym | More Synonyms |
| Description | GSK 1562590 hydrochloride is a high affinity and selective antagonist of urotensin-II receptor (UT), with pKis of 9.14-9.66 for mammalian recombinant (mouse, rat, cat, monkey, human) and native UT[1]. |
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| Related Catalog | |
| References |
| Molecular Formula | C30H31Cl3N4O4 |
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| Molecular Weight | 617.95 |
| Exact Mass | 616.141113 |
| InChIKey | XTVXEMMIPYMBLL-UHFFFAOYSA-N |
| SMILES | CN(C(=O)CN1C(=O)COc2cc(Cl)c(Cl)cc21)C(CN1CCCC1)c1ccc(-c2cccc(C(N)=O)c2)cc1.Cl |
| 4H-1,4-Benzoxazine-4-acetamide, N-[(1R)-1-[3'-(aminocarbonyl)[1,1'-biphenyl]-4-yl]-2-(1-pyrrolidinyl)ethyl]-6,7-dichloro-2,3-dihydro-N-methyl-3-oxo-, hydrochloride (1:1) |
| 4'-[(1R)-1-{[(6,7-Dichloro-3-oxo-2,3-dihydro-4H-1,4-benzoxazin-4-yl)acetyl](methyl)amino}-2-(1-pyrrolidinyl)ethyl]-3-biphenylcarboxamide hydrochloride (1:1) |