TAK-615 structure
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Common Name | TAK-615 | ||
|---|---|---|---|---|
| CAS Number | 1664335-55-0 | Molecular Weight | 419.452 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C25H22FNO4 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of TAK-615TAK-615 (TAK615) is a potent, selective, negative allosteric modulator (NAM) of the LPA1 receptor, partially inhibits the LPA response with IC50 of 91 nM (60% at 10 uM) in calcium mobilisation assays. |
| Name | TAK-615 |
|---|
| Description | TAK-615 (TAK615) is a potent, selective, negative allosteric modulator (NAM) of the LPA1 receptor, partially inhibits the LPA response with IC50 of 91 nM (60% at 10 uM) in calcium mobilisation assays. |
|---|---|
| References | References 1. Ellery J, et al. Eur J Pharmacol. 2018 May 26;833:8-15. View Related Products by Target Lysophospholipid Receptor |
| Molecular Formula | C25H22FNO4 |
|---|---|
| Molecular Weight | 419.452 |
| InChIKey | LEZVXIZCJXKBJY-UHFFFAOYSA-N |
| SMILES | O=C(O)c1ccc(CN(CC2CC2)C(=O)c2ccc(Oc3ccccc3F)cc2)cc1 |