ZEN-3862

Modify Date: 2024-01-14 11:10:14

ZEN-3862 structure	Common Name	ZEN-3862
	CAS Number	1952264-33-3	Molecular Weight	340.35
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₁₉H₁₇FN₂O₃	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of ZEN-3862

ZEN-3862 is a BET inhibitor with IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively. ZEN-3862 can be used to form PROTACs to induce degradation of BRD4[1].

Name	ZEN-3862

Description	ZEN-3862 is a BET inhibitor with IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively. ZEN-3862 can be used to form PROTACs to induce degradation of BRD4[1].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> Epigenetics >> Epigenetic Reader Domain
Target	BRD4 (BD1):0.16 μM (IC50) BRD4 (BD2):0.13 μM (IC50)
References	[1]. Kharenko OA, et al. Design and Characterization of Novel Covalent Bromodomain and Extra-Terminal Domain (BET) Inhibitors Targeting a Methionine. J Med Chem. 2018 Sep 27;61(18):8202-8211.

Molecular Formula	C₁₉H₁₇FN₂O₃
Molecular Weight	340.35

Hazard Codes	Xi

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Shanghai Nianxing Industrial Co., Ltd
China
Product Name: ZEN-3862
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Purity: 98.0%
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The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.