BLU-782

Modify Date: 2024-04-05 07:11:20

BLU-782 Structure
BLU-782 structure
Common Name BLU-782
CAS Number 2141955-96-4 Molecular Weight 562.70
Density N/A Boiling Point N/A
Molecular Formula C31H42N6O4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of BLU-782


ALK2-IN-1 is a activin receptor-like kinase-2 (ALK2) inhibitor extracted from patent WO2017181117A1, Compound 876, has an IC50 of <10 nM[1].

 Names

Name ALK2-IN-1

 BLU-782 Biological Activity

Description ALK2-IN-1 is a activin receptor-like kinase-2 (ALK2) inhibitor extracted from patent WO2017181117A1, Compound 876, has an IC50 of <10 nM[1].
Related Catalog
Target

IC50: <10 nM (ALK2)[1]

References

[1]. Natasja Brooijmans, et al. Inhibitors of activin receptor-like kinase. WO2017181117A1.

 Chemical & Physical Properties

Molecular Formula C31H42N6O4
Molecular Weight 562.70