BAY 6035
Modify Date: 2024-09-18 14:34:28
BAY 6035 structure
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Common Name | BAY 6035 | ||
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| CAS Number | 2247890-13-5 | Molecular Weight | 396.48 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C22H28N4O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of BAY 6035BAY-6035 is a potent, selective and substrate-competitive inhibitor of SMYD3. BAY-6035 inhibits methylation of MEKK2 peptide with an IC50 of 88 nM[1]. |
| Name | BAY-6035 |
|---|
| Description | BAY-6035 is a potent, selective and substrate-competitive inhibitor of SMYD3. BAY-6035 inhibits methylation of MEKK2 peptide with an IC50 of 88 nM[1]. |
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| Related Catalog | |
| Target |
SMYD3:88 nM (IC50) |
| In Vitro | BAY-6035 inhibits in vitro methylation of MEKK2 peptide with an IC50 of 88 nM and has more than 100-fold selectivity over other histone methyltransferases[1]. BAY-6035 inhibits the methylation of MEKK2 in cells with an IC50 of 70 nM[1]. |
| References |
| Molecular Formula | C22H28N4O3 |
|---|---|
| Molecular Weight | 396.48 |