GSK9311 hydrochloride
Modify Date: 2024-01-12 00:37:27
GSK9311 hydrochloride structure
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Common Name | GSK9311 hydrochloride | ||
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| CAS Number | 2253733-09-2 | Molecular Weight | 474.00 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C24H32ClN5O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of GSK9311 hydrochlorideGSK9311 hydrochloride, a less active analogue of GSK6853, can be used as a negative control. GSK9311 hydrochloride inhibits BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively[1]. |
| Name | GSK9311 hydrochloride |
|---|
| Description | GSK9311 hydrochloride, a less active analogue of GSK6853, can be used as a negative control. GSK9311 hydrochloride inhibits BRPF bromodomain with pIC50 values of 6.0 and 4.3 for BRPF1 and BRPF2, respectively[1]. |
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| Related Catalog | |
| Target |
BRPF1:6.0 (pIC50) BRPF2:4.3 (pIC50) |
| In Vitro | GSK6853 is a potent (300 pM), soluble, cell active (20 nM), and highly selective inhibitor of the BRPF1 bromodomain, and demonstrates properties suitable for cellular and in vivo studies. GSK6853 is a less active analogue of GSK6853 in which the 5-amide is alkylated[1]. |
| References |
| Molecular Formula | C24H32ClN5O3 |
|---|---|
| Molecular Weight | 474.00 |