Adenosine receptor inhibitor 2

Modify Date: 2024-04-03 23:46:00

Adenosine receptor inhibitor 2 structure	Common Name	Adenosine receptor inhibitor 2
	CAS Number	2550401-76-6	Molecular Weight	406.28
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₁₇H₂₀BrN₅O₂	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of Adenosine receptor inhibitor 2

Adenosine receptor inhibitor 2 (compound 14b) is a potent AR (adenosine receptor) inhibitor. Adenosine receptor inhibitor 2 shows dual affinity toward A1/A2A ARs with higher affinity for the A1- than the A2AAR. Adenosine receptor inhibitor 2 has Ki values of 52.2 nM for the A1AR and 167 nM for the A2AAR[1].

Name	Adenosine receptor inhibitor 2

Description	Adenosine receptor inhibitor 2 (compound 14b) is a potent AR (adenosine receptor) inhibitor. Adenosine receptor inhibitor 2 shows dual affinity toward A1/A2A ARs with higher affinity for the A1- than the A2AAR. Adenosine receptor inhibitor 2 has Ki values of 52.2 nM for the A1AR and 167 nM for the A2AAR[1].
Related Catalog	Research Areas >> Inflammation/Immunology Signaling Pathways >> GPCR/G Protein >> Adenosine Receptor
Target	A1AR:52.2 ± 8.5 nM (Ki) A2AR:167 ± 22 nM (Ki) hA2B:>1000 nM (Ki) Adenosine A3 receptor:>1000 nM (Ki)
References	[1]. Załuski M, et al. 8-Benzylaminoxanthine scaffold variations for selective ligands acting on adenosine A2A receptors. Design, synthesis and biological evaluation. Bioorg Chem. 2020 Aug;101:104033.

Molecular Formula	C₁₇H₂₀BrN₅O₂
Molecular Weight	406.28

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.

Adenosine receptor inhibitor 2

Use of Adenosine receptor inhibitor 2

Names

Adenosine receptor inhibitor 2 Biological Activity

Chemical & Physical Properties

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.