norastemizole
Modify Date: 2025-08-26 16:22:10
norastemizole structure
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Common Name | norastemizole | ||
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| CAS Number | 75970-99-9 | Molecular Weight | 324.40 | |
| Density | 1.28g/cm3 | Boiling Point | 519.8ºC at 760 mmHg | |
| Molecular Formula | C19H21FN4 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 268.2ºC | |
Use of norastemizoleTecastemizole (Norastemizole), a major metabolite of Astemizole, is a potent and selective H1 receptor antagonist. Tecastemizole shows anti-inflammatory activities[1]. |
| Name | 1-[(4-fluorophenyl)methyl]-N-piperidin-4-ylbenzimidazol-2-amine |
|---|---|
| Synonym | More Synonyms |
| Description | Tecastemizole (Norastemizole), a major metabolite of Astemizole, is a potent and selective H1 receptor antagonist. Tecastemizole shows anti-inflammatory activities[1]. |
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| Related Catalog | |
| References |
| Density | 1.28g/cm3 |
|---|---|
| Boiling Point | 519.8ºC at 760 mmHg |
| Molecular Formula | C19H21FN4 |
| Molecular Weight | 324.40 |
| Flash Point | 268.2ºC |
| Exact Mass | 324.17500 |
| PSA | 45.11000 |
| LogP | 3.13830 |
| Index of Refraction | 1.658 |
| InChIKey | SFOVDSLXFUGAIV-UHFFFAOYSA-N |
| SMILES | Fc1ccc(Cn2c(NC3CCNCC3)nc3ccccc32)cc1 |
| Storage condition | 2-8°C |
| Precursor 10 | |
|---|---|
| DownStream 2 | |
![4-[[1-[(4-FLUOROPHENYL)-METHYL]-1H-BENZIMIDAZOLE-2-YL]AMINO]-1-PIPERIDINECARBOXYLIC ACID ETHYL ESTER Structure](https://image.chemsrc.com/caspic/340/84501-68-8.png)
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CAS#:73734-07-3![1-[(4-Fluorophenyl)methyl]-N-[1-[2-(2-pyridinyl)ethyl]-4-piperidinyl]-1H-benzimidazol-2-amine structure](https://image.chemsrc.com/caspic/486/73735-69-0.png)
CAS#:73735-69-0|
Name: Antimalarial activity against Plasmodium falciparum 3D7 infected in ARh+ human erythr...
Source: ChEMBL
Target: Plasmodium falciparum
External Id: CHEMBL4180222
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Name: Antimalarial activity against Plasmodium falciparum 3D7 infected in ARh+ human erythr...
Source: ChEMBL
Target: Plasmodium falciparum
External Id: CHEMBL4180223
|
|
Name: Inhibition of human Potassium channel HERG expressed in mammalian cells
Source: ChEMBL
Target: Potassium voltage-gated channel subfamily H member 2
External Id: CHEMBL766814
|
|
Name: Antimalarial activity against Plasmodium falciparum 3D7 infected in ARh+ human erythr...
Source: ChEMBL
Target: Plasmodium falciparum
External Id: CHEMBL4180219
|
|
Name: Antimalarial activity against Plasmodium falciparum 3D7 infected in ARh+ human erythr...
Source: ChEMBL
Target: Plasmodium falciparum
External Id: CHEMBL4180220
|
|
Name: Antimalarial activity against Plasmodium falciparum 3D7 infected in ARh+ human erythr...
Source: ChEMBL
Target: Plasmodium falciparum
External Id: CHEMBL4180221
|
|
Name: Inhibition of human ERG expressed in CHO cells by whole cell patch clamp technique
Source: ChEMBL
Target: Potassium voltage-gated channel subfamily H member 2
External Id: CHEMBL954102
|
|
Name: Enzymatic assay of human HDAC6 with commercial peptide substrate
Source: ChEMBL
Target: Histone deacetylase 6
External Id: CHEMBL4808149
|
|
Name: Enzymatic assay of human HDAC6 with custom peptide substrate
Source: ChEMBL
Target: Histone deacetylase 6
External Id: CHEMBL4808150
|
|
Name: Inhibition of human ERG channel in HEK293 cells by voltage-clamp method
Source: ChEMBL
Target: Potassium voltage-gated channel subfamily H member 2
External Id: CHEMBL1036648
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| T 1348 |
| Tetemizole |
| Soltara |
| Norastemizole |