Cazpaullone

Modify Date: 2024-01-10 11:29:58

Cazpaullone Structure
Cazpaullone structure
Common Name Cazpaullone
CAS Number 914088-64-5 Molecular Weight 274.27700
Density 1.49±0.1 g/cm3 (20 °C, 760 mmHg) Boiling Point 680.7±50.0 °C (760 mmHg)
Molecular Formula C16H10N4O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Cazpaullone


Cazpaullone is a glycogen synthase kinase-3 (GSK-3) inhibitor. Cazpaullone can activate pancreatic beta cell protection and replication. Cazpaullone can be used for the research of diabetes[1].

 Names

Name Pyrido[3',2':2,3]azepino[4,5-b]indole-9-carbonitrile, 5,6,7,12-tetrahydro-6-oxo
Synonym More Synonyms

 Cazpaullone Biological Activity

Description Cazpaullone is a glycogen synthase kinase-3 (GSK-3) inhibitor. Cazpaullone can activate pancreatic beta cell protection and replication. Cazpaullone can be used for the research of diabetes[1].
Related Catalog
References

[1]. Stukenbrock H, et al. 9-cyano-1-azapaullone (cazpaullone), a glycogen synthase kinase-3 (GSK-3) inhibitor activating pancreatic beta cell protection and replication. J Med Chem. 2008 Apr 10;51(7):2196-207.  

 Chemical & Physical Properties

Density 1.49±0.1 g/cm3 (20 °C, 760 mmHg)
Boiling Point 680.7±50.0 °C (760 mmHg)
Molecular Formula C16H10N4O
Molecular Weight 274.27700
Exact Mass 274.08500
PSA 81.57000
LogP 2.73418

 Synonyms

CAZPAULLONE
Cazpaullone