ISAM 140
Modify Date: 2024-01-10 20:58:07
ISAM 140 structure
|
Common Name | ISAM 140 | ||
|---|---|---|---|---|
| CAS Number | 932191-62-3 | Molecular Weight | 337.37 | |
| Density | 1.3±0.1 g/cm3 | Boiling Point | 503.0±60.0 °C at 760 mmHg | |
| Molecular Formula | C19H19N3O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 258.0±32.9 °C | |
Use of ISAM 140ISAM-140 (22b) is a potent and highly selective A2B adenosine receptor antagonist with a Ki of 3.49 nM[1]. |
| Name | ISAM-140 |
|---|---|
| Synonym | More Synonyms |
| Description | ISAM-140 (22b) is a potent and highly selective A2B adenosine receptor antagonist with a Ki of 3.49 nM[1]. |
|---|---|
| Related Catalog | |
| Target |
hA2B:3.49 nM (Ki) |
| In Vitro | ISAM-140 (22b) (0.1-100 µM) inhibits NECA (5'-N-ethylcarboxamido adenosine)-stimulated cAMP accumulation[1]. ISAM-140 shows a KB value of 27.00 nM[1]. |
| References |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 503.0±60.0 °C at 760 mmHg |
| Molecular Formula | C19H19N3O3 |
| Molecular Weight | 337.37 |
| Flash Point | 258.0±32.9 °C |
| Exact Mass | 337.142639 |
| LogP | 4.42 |
| Vapour Pressure | 0.0±1.3 mmHg at 25°C |
| Index of Refraction | 1.659 |
| Isopropyl 4-(2-furyl)-2-methyl-4,10-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate |
| Isopropyl 4-(2-furyl)-2-methyl-1,4-dihydropyrimido[1,2-a]benzimidazole-3-carboxylate |
| Pyrimido[1,2-a]benzimidazole-3-carboxylic acid, 4-(2-furanyl)-1,4-dihydro-2-methyl-, 1-methylethyl ester |
| Pyrimido[1,2-a]benzimidazole-3-carboxylic acid, 4-(2-furanyl)-4,10-dihydro-2-methyl-, 1-methylethyl ester |
| MFCD09438096 |
| 4-(2-Furanyl)-4,10-dihydro-2-methyl-pyrimido[1,2-a]benzimidazole-3-carboxylic acid 1-methylethyl ester |
| ISAM-140 |
| (±)-Isopropyl 4-(Furan-2-yl)-2-methyl-1,4-dihydrobenzo-[4,5]imidazo[1,2-a]pyrimidine-3-carboxylate |