(Lys4)-Sarafotoxin C acetate salt

• 常用名: (Lys4)-Sarafotoxin C acetate salt
• 英文名: (Lys4)-Sarafotoxin C acetate salt
• CAS号: 1219444-22-0
• 分子量: 2529.823
• 密度: 1.3±0.1 g/cm3
• 沸点: 2622.4±65.0 °C at 760 mmHg
• 分子式: C₁₀₅H₁₅₃N₂₇O₃₆S₅
• 熔点: N/A
• 闪点: 1539.8±34.3 °C

(Lys4)-Sarafotoxin C acetate salt用途

[Lys4]Sarafotoxin S6c,一种Sarafotoxix类似物,是内皮素受体的有效和部分激动剂。[Lys4]Sarafotoxin S6c引起猪冠状动脉收缩,EC50为1.5 nM[1]。

(Lys4)-Sarafotoxin C acetate salt名称

• 英文名: (Lys4)-Sarafotoxin C acetate salt

(Lys4)-Sarafotoxin C acetate salt生物活性

• 描述: [Lys4]Sarafotoxin S6c,一种Sarafotoxix类似物,是内皮素受体的有效和部分激动剂。[Lys4]Sarafotoxin S6c引起猪冠状动脉收缩,EC50为1.5 nM[1]。
• 相关类别:
  研究领域 >> 心血管疾病
  信号通路 >> G 蛋白偶联受体/G 蛋白 >> 内皮素受体
• 体外研究: [Lys4]Sarafotoxin S6c与Sarafotoin S6c[1]具有同等的亲和力。

(Lys4)-Sarafotoxin C acetate salt物理化学性质

• 密度: 1.3±0.1 g/cm3
• 沸点: 2622.4±65.0 °C at 760 mmHg
• 分子式: C₁₀₅H₁₅₃N₂₇O₃₆S₅
• 分子量: 2529.823
• 闪点: 1539.8±34.3 °C
• 精确质量: 2527.957520
• LogP: -5.95
• 蒸汽压: 0.0±0.3 mmHg at 25°C
• 折射率: 1.558

(Lys4)-Sarafotoxin C acetate salt英文别名

• MFCD00133969
• L-Tryptophan, N-[[(1R,4S,7S,10S,13S,16S,19S,22S,25R,28S,31R,36R,39S,42S,45S)-31-amino-22-(4-aminobutyl)-42-(2-amino-2-oxoethyl)-4,7-bis(2-carboxyethyl)-10,19-bis(carboxymethyl)-13,28-bis[(1R)-1-hydroxyethyl]-45-(2-methylpropyl)-16-[2-(methylthio)ethyl]-3,6,9,12,15,18,21,24,27,30,38,41,44,47-tetradecaoxo-39-(phenylmethyl)-33,34,49,50-tetrathia-2,5,8,11,14,17,20,23,26,29,37,40,43,46-tetradecaazabicyclo[23.22.4]henpentacont-36-yl]carbonyl]-L-h
• N-({(1R,4S,7S,10S,13S,16S,19S,22S,25R,28S,31R,36R,39S,42S,45S)-31-Amino-22-(4-aminobutyl)-42-(2-amino-2-oxoethyl)-39-benzyl-4,7-bis(2-carboxyethyl)-10,19-bis(carboxymethyl)-13,28-bis[(1R)-1-hydroxyethyl]-45-isobutyl-16-[2-(methylsulfanyl)ethyl]-3,6,9,12,15,18,21,24,27,30,38,41,44,47-tetradecaoxo-33,34,49,50-tetrathia-2,5,8,11,14,17,20,23,26,29,37,40,43,46-tetradecaazabicyclo[23.22.4]henpentacont-36-yl}carbonyl)-L-histidyl-L-glutaminyl-L-alp