强啡肽A结构式
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常用名 | 强啡肽A | 英文名 | Dynorphin A trifluoroacetate salt |
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CAS号 | 80448-90-4 | 分子量 | 2147.484 | |
密度 | 1.5±0.1 g/cm3 | 沸点 | N/A | |
分子式 | C99H155N31O23 | 熔点 | N/A | |
MSDS | 中文版 美版 | 闪点 | N/A |
Dynorphin A as a potential endogenous ligand for four members of the opioid receptor gene family.
J. Pharmacol. Exp. Ther. 286 , 136-141, (1998) Dynorphin A is an endogenous opioid peptide that activates the kappa opioid receptor (KOR) with high potency. Some studies also showed that the distribution and functional activity of dynorphin A are not completely correlated with those of KOR, suggesting tha... |
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Structure-activity relationship studies of dynorphin A and related peptides.
Peptides 19 , 1277-1292, (1998) An up-to-date review is presented covering all the available information concerning the isolation, discovery, synthesis, conformation, receptor binding characteristics, pharmacological properties and SAR studies of dynorphin A and related peptides. The potent... |
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The kappa opioid receptor and dynorphin co-localize in vasopressin magnocellular neurosecretory neurons in guinea-pig hypothalamus.
Neuroscience 96 , 373-383, (2000) The relationship between the cloned kappa opioid receptor, dynorphin, and the neurohypophysial hormones vasopressin and oxytocin was analysed in the guinea-pig hypothalamic magnocellular neurosecretory neurons. This analysis was performed in order to understa... |