N-Fmoc-D-1,2,3,4-四氢异喹啉-3-羧酸
N-Fmoc-D-1,2,3,4-四氢异喹啉-3-羧酸结构式
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常用名 | N-Fmoc-D-1,2,3,4-四氢异喹啉-3-羧酸 | 英文名 | Fmoc-D-Tic-OH |
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| CAS号 | 130309-33-0 | 分子量 | 399.439 | |
| 密度 | 1.3±0.1 g/cm3 | 沸点 | 629.9±55.0 °C at 760 mmHg | |
| 分子式 | C25H21NO4 | 熔点 | 160-164 °C | |
| MSDS | 中文版 美版 | 闪点 | 334.7±31.5 °C |
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Bradykinin receptor antagonists containing N-substituted amino acids: in vitro and in vivo B(2) and B(1) receptor antagonist activity.
J. Med. Chem. 39 , 1472, (1996) We report a systematic probing of the structural requirements of the bradykinin (BK) type 2 (B(2)) receptor for antagonist activity by incorporating N-alkyl-amino acid residues at positions 7 and 8 of a potent antagonist sequence. Compound 1 (D-Arg(0)-Arg(1)-... |
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Design and synthesis of new linear and cyclic bradykinin antagonists.
J. Med. Chem. 39 , 2095, (1996) We report here on the synthesis and pharmacological properties of a new series of small linear and cyclic peptides derived from the five C-terminal amino acid residues of second-generation bradykinin receptor antagonists. Variations of the two first residues ... |
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