946578-00-3

• 常用中文名：氟啶虫胺腈
• 常用英文名：Sulfoxaflor
• CAS号：946578-00-3
• 分子式：C₁₀H₁₀F₃N₃OS
• 分子量：277.26600
• 相关类别： 化学农药原药 杀虫剂 有机氯杀虫剂
• 发布时间：2018-05-27 08:00:00
• 更新时间：2026-07-17 00:16:09
• Sulfoxaflor 是磺胺嘧啶的杀虫剂,是 nAChR1 和 nAChR2 亚型的激动剂。Sulfoxaflor 可用于控制食树性昆虫,如桃蚜,棉蚜,烟粉虱和褐飞虱。

名称

• 中文名: 氟啶虫胺腈
• 英文名: sulfoxaflor
• 中文别名: 正己烷中氟啶虫胺腈溶液标准物质; 氟啶虫胺腈溶液, 100PPM; 啶虫胺腈; 甲醇中氟啶虫胺腈溶液标准物质; 氟啶虫胺腈(砜虫啶); 砜虫啶/氟啶虫胺腈; 氟啶虫胺腈,1000PPM; 乙腈中氟啶虫胺腈溶液标准物质; 磺草胺(2- 甲基 -13C, 氰胺 -15N2; 氟啶虫胺腈溶液; 氟啶虫胺腈水分散粒剂WDG; 砜虫啶; 亚胺 -15N,); 甲基[1-(2-三氟甲基吡啶-5-基)乙基]-N-氰基亚磺酰亚胺; 氟啶虫胺腈溶液, 1000PPM; 磺草胺(氰基 -13C; 亚砜草胺(100UG/ML 在甲烷中的混合物; 乙腈中氟啶虫胺腈; [1-[6-(三氟甲基）吡啶-3-基]乙基]甲基(氧)-λ4-巯基氨腈; 亚砜草胺; 氟啶虫胺腈,1MG/ML甲醇溶液
• 英文别名: Sulfoxaflor , WDG; l^{6}-sulfanylidene]cyanamide; Sulfoxaflor solution,1000ppm; Transform 50 WG (Sulfoxaflor WDG); Sulfoxaflor solution; Sulfoxaflor(mixture of isomers); [(Ξ)-methyl(oxo){(1Ξ)-1-[6-(trifluoromethyl)pyridin-3-yl]ethyl}-λ6-sulfanylidene]cyanamide; [6-[trifluoromethylpyridin-3-yl]ethyl](methyl)oxido-lambda4-sulphanylidene-cyanamide; Sulfoxaflor@1000 μg/mL in Acetonitrile; Cyanamide,N-[methyloxido[1-[6-(trifluoromethyl)-3-pyridinyl]ethyl]-l4-sulfanylidene]; Cyamide,N-[methyloxido[1-[6-(trifluoromethyl)-3-pyridinyl]ethyl]-l4-sulfanylidene]; Sulfoxaflo; N-(methyloxido(1-(6-(trifluoromethyl)-3-pyridinyl)ethyl)-lambda4-sulfanylidene)cyanamide; [methyl(oxo){1-[6-(trifluoromethyl)-3-pyridyl]ethyl}-λ6-sulfanylidene]cyanamide; [methyl-oxo-[1-[6-(trifluoromethyl)pyridin-3-yl]ethyl]-; Sulfoxaflor WDG; Sulfoxaflor 100 μg/ml Acetonitrile; [methyl-oxo-[1-[6-(trifluoromethyl)pyridin-3-yl]ethyl]-λ⁶-sulfanylidene]cyanamide; GF 2372; Sulfoxaflor@100 μg/mL in Methanol; GF 2032; Sulfoxaflor 100 μg/ml Acetone; Methyl[1-(2-trifluoromethylpyridin-5-yl)ethyl]-N-cyanosulfoximine; Cyanamide, N-[methyloxido[1-[6-(trifluoromethyl)-3-pyridinyl]ethyl]-λ4-sulfanylidene]; Sulfoxaflor 100 μg/mL in Acetonitrile; SULFANONE; [methyl(oxido){1-[6-(trifluoromethyl)pyridin-3-yl]ethyl}-lambda~4~-sulfanylidene]cyanamide; Sulfoximine,Inhibitor,median,unpaired,insecticide,dorsal,nAChR1,Sulfoxaflor,nAChR2,Nicotinic acetylcholine rectors,inhibit,nAChR; N-[methyloxido[1-[6-(trifluoromethyl)-3-pyridinyl]ethyl]-λ4-sulfanylidene]cyanamide; Sulfoxaflor in Acetonitrile; Sulfoxaflor [ISO]; (CYANOIMINO)(METHYL){1-[6-(TRIFLUOROMETHYL)PYRIDIN-3-YL]ETHYL}-Λ⁶; C17015000 Sulfoxaflor; Transform 50 WG; 13c,); (cyanoimino)(methyl){1-[6-(trifluoromethyl)pyridin -3-yl]ethyl}-lambda6-sulfanone; [methyl(oxido){1-[6-(trifluoromethyl)pyridin-3-yl]ethyl}-lam; XDE 208; Transfmer (Sulfoxaflor) 50 WG; Transform; Sulfoxaflor 100 μg/ml Methanol; Transform WG New Insecticide Label for Cotton

物化性质

• 密度: 1.34g/cm3
• 沸点: 363.8ºC at 760 mmHg
• 分子式: C₁₀H₁₀F₃N₃OS
• 分子量: 277.26600
• 闪点: 173.8ºC
• 精确质量: 277.05000
• PSA: 74.49000
• LogP: 3.60598
• 折射率: 1.519
• 储存条件: -20°C， 密封， 干燥

生物活性

• 描述: Sulfoxaflor 是磺胺嘧啶的杀虫剂,是 nAChR1 和 nAChR2 亚型的激动剂。Sulfoxaflor 可用于控制食树性昆虫,如桃蚜,棉蚜,烟粉虱和褐飞虱。
• 相关类别:
  信号通路 >> 跨膜转运 >> 胆碱受体
  信号通路 >> 神经信号通路 >> 胆碱受体
  研究领域 >> 神经疾病
• 参考文献:

  [1]. Jean-Noël Houchat, et al. Mode of Action of Sulfoxaflor on α-bungarotoxin-insensitive nAChR1 and nAChR2 Subtypes: Inhibitory Effect of Imidacloprid. Neurotoxicology. 2019 Sep;74:132-138.

安全

• 危害码 (欧洲): Xi

合成路线

946577-99-7 74-88-4 ~60% 946578-00-3

文献：Dow AgroSciences, LLC Patent: US2010/168177 A1, 2010 ; Location in patent: Page/Page column 5-6 ;

1049684-75-4 ~90% 946578-00-3

文献：DOW AGROSCIENCES LLC Patent: WO2008/97235 A1, 2008 ; Location in patent: Page/Page column 18-20 ;

1046119-63-4 ~65% 946578-00-3

文献：Dow AgroSciences LLC Patent: US2008/207910 A1, 2008 ; Location in patent: Page/Page column 6; 7 ;

946577-96-4 ~% 946578-00-3

文献：Dow AgroSciences LLC; Babcock, Jonathan M.; Young, Catherine D.; King, James E.; Kubiszak, Mary E. Patent: US2013/288897 A1, 2013 ;

946577-97-5 ~% 946578-00-3

文献：Dow AgroSciences LLC; Babcock, Jonathan M.; Young, Catherine D.; King, James E.; Kubiszak, Mary E. Patent: US2013/288897 A1, 2013 ;

386715-33-9 ~% 946578-00-3

文献：Dow AgroSciences LLC; Babcock, Jonathan M.; Young, Catherine D.; King, James E.; Kubiszak, Mary E. Patent: US2013/288897 A1, 2013 ;