arg-pro-pro-gly-phe-ser-pro-leu acetate salt结构式
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常用名 | arg-pro-pro-gly-phe-ser-pro-leu acetate salt | 英文名 | arg-pro-pro-gly-phe-ser-pro-leu acetate salt |
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| CAS号 | 115035-45-5 | 分子量 | 930.06 | |
| 密度 | N/A | 沸点 | N/A | |
| 分子式 | C43H67N11O12 | 熔点 | N/A | |
| MSDS | 美版 | 闪点 | N/A |
用途Des-Arg9-[Leu8]-Bradykinin acetate 是有效的 缓激肽受体1 (B1R) 拮抗剂。Des-Arg9-[Leu8]-Bradykinin acetate 可用于肾纤维化研究。 |
| 英文名 | arg-pro-pro-gly-phe-ser-pro-leu acetate salt |
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| 英文别名 | 更多 |
| 描述 | Des-Arg9-[Leu8]-Bradykinin acetate 是有效的 缓激肽受体1 (B1R) 拮抗剂。Des-Arg9-[Leu8]-Bradykinin acetate 可用于肾纤维化研究。 |
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| 相关类别 | |
| 靶点实验 |
IC50: B1R[1] |
| 参考文献 |
| 分子式 | C43H67N11O12 |
|---|---|
| 分子量 | 930.06 |
| 精确质量 | 929.49700 |
| PSA | 360.08000 |
| LogP | 0.84570 |
| InChIKey | XBFMNOKHQZCARQ-XXZMQFNDSA-N |
| SMILES | CC(=O)O.CC(C)CC(NC(=O)C1CCCN1C(=O)C(CO)NC(=O)C(Cc1ccccc1)NC(=O)CNC(=O)C1CCCN1C(=O)C1CCCN1C(=O)C(N)CCCN=C(N)N)C(=O)O |
| 个人防护装备 | Eyeshields;Gloves;type N95 (US);type P1 (EN143) respirator filter |
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| 危险品运输编码 | NONH for all modes of transport |
| WGK德国 | 3 |
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Upregulation of B1 receptor mediating des-Arg9-BK-induced rat paw oedema by systemic treatment with bacterial endotoxin.
Br. J. Pharmacol. 117 , 793-798, (1996) 1. The effect of pretreatment with bacterial endotoxin (LPS, 10 micrograms, i.v., 24 h) on the bradykinin B1 and B2 receptor-induced oedema in the rat paw, and the interaction of B1-mediated responses... |
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Angiotensin II type 2 receptor expression after vascular injury: differing effects of angiotensin-converting enzyme inhibition and angiotensin receptor blockade.
Hypertension 48 , 942-949, (2006) It has been suggested that the effects of angiotensin II type 1 receptor (AT1R) blockers are in part because of angiotensin II type 2 receptor (AT2R) signaling. Interactions between the AT2R and kinin... |
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The role of kinin B1 receptors in the nociception produced by peripheral protein kinase C activation in mice.
Neuropharmacology 54 , 597-604, (2008) The peripheral injection of phorbol myristate acetate (PMA) into the mouse paw induces nociception mediated through activation of protein kinase C (PKC). In the present study, we examine the contribut... |
| arg-pro-pro-gly-phe-ser-pro-leu acoh 3h2o |