4-Bromoindole

4-Bromoindole Structure
4-Bromoindole structure
Common Name 4-Bromoindole
CAS Number 52488-36-5 Molecular Weight 196.044
Density 1.7±0.1 g/cm3 Boiling Point 316.9±15.0 °C at 760 mmHg
Molecular Formula C8H6BrN Melting Point 17 °C
MSDS Chinese USA Flash Point 145.5±20.4 °C
Symbol GHS07
GHS07
Signal Word Warning

A concise and scalable strategy for the total synthesis of dictyodendrin B based on sequential C-H functionalization.

Angew. Chem. Int. Ed. Engl. 54(18) , 5451-5, (2015)

A sequential CH functionalization strategy for the synthesis of the marine alkaloid dictyodendrin B is reported. Our synthesis begins from commercially available 4-bromoindole and involves six direct functionalizations around the heteroarene core as part of ...

Applications of vinylogous Mannich reactions. Total syntheses of the Ergot alkaloids rugulovasines A and B and setoclavine.

J. Am. Chem. Soc. 123(25) , 5918-24, (2001)

Concise syntheses of the Ergot alkaloids rugulovasine A (3a), rugulovasine B (3b), and setoclavine (2) have been completed by strategies that feature inter- and intramolecular vinylogous Mannich reactions as the key steps. Thus, the first synthesis of 3a,b co...

Optically active total synthesis of clavicipitic acid. Yokoyama Y, et al.

J. Org. Chem. 60(6) , 1486-1487, (1995)

Metal-halogen exchange of bromoindoles. A route to substituted indoles. Moyer MP, et al.

J. Org. Chem. 51(26) , 5106-5110, (1986)