A2A receptor antagonist 1

Modify Date: 2024-01-10 19:20:36

A2A receptor antagonist 1 structure	Common Name	A2A receptor antagonist 1
	CAS Number	443103-97-7	Molecular Weight	309.3
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₁₆H₁₂FN₅O	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of A2A receptor antagonist 1

A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.

Name	A2A receptor antagonist 1

Description	A2A receptor antagonist 1 is an antagonist of both adenosine A2A receptor and A1 receptor with Kis of 4 and 264 nM, respectively.
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Adenosine Receptor Research Areas >> Cancer Research Areas >> Neurological Disease
Target	Ki: 4 nM (adenosine A2A receptor), 264 nM (A1 receptor)[1]
References	[1]. Gillespie RJ, et al. Antagonists of the human adenosine A2A receptor. Part 3: Design and synthesis of pyrazolo[3,4-d]pyrimidines, pyrrolo[2,3-d]pyrimidines and 6-arylpurines. Bioorg Med Chem Lett. 2008 May 1;18(9):2924-9.

Molecular Formula	C₁₆H₁₂FN₅O
Molecular Weight	309.3
Storage condition	-20℃