Dopamine D2 receptor antagonist-1

Modify Date: 2024-01-12 09:18:40

Dopamine D2 receptor antagonist-1 Structure
Dopamine D2 receptor antagonist-1 structure
Common Name Dopamine D2 receptor antagonist-1
CAS Number 1055411-77-2 Molecular Weight 259.37
Density N/A Boiling Point N/A
Molecular Formula C14H17N3S Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Dopamine D2 receptor antagonist-1


Dopamine D2 receptor antagonist-1 is a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R) with sub-mM affinity[1].

 Names

Name Dopamine D2 receptor antagonist-1

 Dopamine D2 receptor antagonist-1 Biological Activity

Description Dopamine D2 receptor antagonist-1 is a negative allosteric modulator (NAM) of the dopamine D2 receptor (D2R) with sub-mM affinity[1].
Related Catalog
Target

D2R[1]

References

[1]. Fyfe TJ, et al. Subtle modifications to a thieno[2,3-d]pyrimidine scaffold yield negative allosteric modulators and agonists of the dopamine D2 receptor. Eur J Med Chem. 2019 Apr 15;168:474-490.

 Chemical & Physical Properties

Molecular Formula C14H17N3S
Molecular Weight 259.37