CCK-B Receptor Antagonist 2

Modify Date: 2025-08-25 12:34:40

CCK-B Receptor Antagonist 2 structure	Common Name	CCK-B Receptor Antagonist 2
	CAS Number	155412-88-7	Molecular Weight	484.55
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₇H₂₈N₆O₃	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of CCK-B Receptor Antagonist 2

CCK-B Receptor Antagonist 2, compound 15b, is a potent and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.43 nM. CCK-B Receptor Antagonist 2 also inhibits gastrin/CCK-A activity with an IC50 of 1.82 μM[1].

Name	CCK-B Receptor Antagonist 2

Description	CCK-B Receptor Antagonist 2, compound 15b, is a potent and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.43 nM. CCK-B Receptor Antagonist 2 also inhibits gastrin/CCK-A activity with an IC50 of 1.82 μM[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Cholecystokinin Receptor Research Areas >> Metabolic Disease
Target	IC50: 0.43 nM (Gastrin/CCK-B); 1.82 μM (Gastrin/CCK-A)[1]
In Vivo	CCK-B Receptor Antagonist 2 (0.1 μmol/kg; intravenous injection) has an inhibition effect on pentagastrin-induced gastric acid secretion in anethsetized rats with an ED50 of 8.3 nmol/kg[1].
References	[1]. Semple G, et al. (3R)-N-(1-(tert-butylcarbonylmethyl)-2,3-dihydro-2-oxo-5-(2-pyridyl)-1H-1,4-benzodiazepin-3-yl)-N'-(3-(methylamino)phenyl)urea (YF476): a potent and orally active gastrin/CCK-B antagonist.J Med Chem. 1997 Jan 31;40(3):331-41.

Molecular Formula	C₂₇H₂₈N₆O₃
Molecular Weight	484.55

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.

Shanghai Nianxing Industrial Co., Ltd
China
Product Name: CCK-B Receptor Antagonist 2
Price: Check
Purity: 98.0%
Delivery: 10 Day
Contact: Yang
Email: sales@echemcloud.com

DC Chemicals Limited
China
Product Name: CCK-B Receptor Antagonist 2
Price: $Inquiry/1g
Purity: 98.0%
Delivery: 3 Day
Contact: Tony Cao
Email: sales@dcchemicals.com

ShangHai DC Chemicals Co.,Ltd
China
Product Name: CCK-B Receptor Antagonist 2
Price: ￥Inquiry/1g
Purity: 98.9%
Delivery: 1 Day
Contact: Tony Lai
Email: order@dcchemicals.com

Get all suppliers and price by the below link:

CCK-B Receptor Antagonist 2 suppliers

Price: ￥4500/5 mg

Reference only. check more CCK-B Receptor Antagonist 2 price

CCK-B Receptor Antagonist 2

Use of CCK-B Receptor Antagonist 2

Names

CCK-B Receptor Antagonist 2 Biological Activity

Chemical & Physical Properties

The content on this webpage is sourced from various professional data sources. If you have any questions or concerns regarding the content, please feel free to contact service1@chemsrc.com.