BET-IN-2

Modify Date: 2024-01-10 15:25:44

BET-IN-2 Structure
BET-IN-2 structure
Common Name BET-IN-2
CAS Number 2104688-91-5 Molecular Weight 363.50
Density N/A Boiling Point N/A
Molecular Formula C23H29N3O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of BET-IN-2


BET-IN-2 is a BET inhibitor with an IC50 of 52 nM for BRD4-BD1.

 Names

Name BET-IN-2

 BET-IN-2 Biological Activity

Description BET-IN-2 is a BET inhibitor with an IC50 of 52 nM for BRD4-BD1.
Related Catalog
Target

BRD4 BD1:52 nM (IC50)

References

[1]. Hu J, et al. Discovery of a series of dihydroquinoxalin-2(1H)-ones as selective BET inhibitors from a dual PLK1-BRD4 inhibitor. Eur J Med Chem. 2017 Sep 8;137:176-195.

 Chemical & Physical Properties

Molecular Formula C23H29N3O
Molecular Weight 363.50