JWG-071
Modify Date: 2024-01-15 11:45:24
JWG-071 structure
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Common Name | JWG-071 | ||
|---|---|---|---|---|
| CAS Number | 2250323-50-1 | Molecular Weight | 612.76 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C34H44N8O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of JWG-071JWG-071 is the first reported kinase-selective chemical probe for ERK5. JWG-071 improves ERK5 activity and BRD4 selectivity. JWG-071 will be a much-needed chemical probe for deconvoluting ERK5 and BRD4 pharmacology[1]. |
| Name | JWG-071 |
|---|
| Description | JWG-071 is the first reported kinase-selective chemical probe for ERK5. JWG-071 improves ERK5 activity and BRD4 selectivity. JWG-071 will be a much-needed chemical probe for deconvoluting ERK5 and BRD4 pharmacology[1]. |
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| Related Catalog | |
| Target |
ERK5:88 nM (IC50) |
| In Vitro | JWG-071 inhibits ERK5 and LRRK2 with IC50 of 88 and 109 nM, respectively[1]. |
| References |
| Molecular Formula | C34H44N8O3 |
|---|---|
| Molecular Weight | 612.76 |