σ1 Receptor/μ Opioid receptor modulator 1

Modify Date: 2024-01-12 10:45:11

σ1 Receptor/μ Opioid receptor modulator 1 structure	Common Name	σ1 Receptor/μ Opioid receptor modulator 1
	CAS Number	2412700-00-4	Molecular Weight	398.51
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₄H₃₁FN₂O₂	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of σ1 Receptor/μ Opioid receptor modulator 1

σ1 Receptor/μ Opioid receptor modulator 1 (Compound 44) is a potent σ1 receptor antagonist and μ opioid receptor agonist with Kis of 1.86 nM and 2.1 nM, respectively.σ1 Receptor/μ Opioid receptor modulator 1 exhibits potent analgesic activity. σ1 Receptor/μ Opioid receptor modulator 1 can be used for the research of neuropathic pain[1].

Name	σ1 Receptor/μ Opioid receptor modulator 1

Description	σ1 Receptor/μ Opioid receptor modulator 1 (Compound 44) is a potent σ1 receptor antagonist and μ opioid receptor agonist with Kis of 1.86 nM and 2.1 nM, respectively.σ1 Receptor/μ Opioid receptor modulator 1 exhibits potent analgesic activity. σ1 Receptor/μ Opioid receptor modulator 1 can be used for the research of neuropathic pain[1].
Related Catalog	Signaling Pathways >> GPCR/G Protein >> Opioid Receptor Signaling Pathways >> Neuronal Signaling >> Opioid Receptor Research Areas >> Neurological Disease Signaling Pathways >> GPCR/G Protein >> Sigma Receptor
References	[1]. Jiaying Xiong, et al. Piperidine propionamide as a scaffold for potent sigma-1 receptor antagonists and mu opioid receptor agonists for treating neuropathic pain. Eur J Med Chem. 2020 Apr 1;191:112144.

Molecular Formula	C₂₄H₃₁FN₂O₂
Molecular Weight	398.51

σ1 Receptor/μ Opioid receptor modulator 1

Use of σ1 Receptor/μ Opioid receptor modulator 1

Names

Biological Activity

Chemical & Physical Properties