lucPpy-IN-1

Modify Date: 2024-04-06 10:56:04

lucPpy-IN-1 Structure
lucPpy-IN-1 structure
Common Name lucPpy-IN-1
CAS Number 546100-66-7 Molecular Weight 409.48
Density 1.410±0.06 g/cm3(Predicted) Boiling Point 312.4±37.0 °C(Predicted)
Molecular Formula C25H23N5O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of lucPpy-IN-1


lucPpy-IN-1 (compound 9) is an ATP-dependent luciferase from Photinus pyralis (lucPpy) inhibitor with an IC50 value of 4.0 µM. lucPpy-IN-1 can be used for the research of target’s druggability[1].

 Names

Name WAY-350568
Synonym More Synonyms

 lucPpy-IN-1 Biological Activity

Description lucPpy-IN-1 (compound 9) is an ATP-dependent luciferase from Photinus pyralis (lucPpy) inhibitor with an IC50 value of 4.0 µM. lucPpy-IN-1 can be used for the research of target’s druggability[1].
Related Catalog
Target

IC50: 4.0 µM (lucPpy)[1]

In Vitro lucPpy-IN-1 (0.1 nM-100 µM) inhibits activity of lucPpy with an IC50 value of 4.0 µM[1].
References

[1]. Auld DS, et al. A basis for reduced chemical library inhibition of firefly luciferase obtained from directed evolution. J Med Chem. 2009 Mar 12;52(5):1450-8.  

 Chemical & Physical Properties

Density 1.410±0.06 g/cm3(Predicted)
Boiling Point 312.4±37.0 °C(Predicted)
Molecular Formula C25H23N5O
Molecular Weight 409.48

 Synonyms

Methanone, [2-(4-methylphenyl)-4-quinolinyl][4-(2-pyrimidinyl)-1-piperazinyl]-