HE-2500 structure
|
Common Name | HE-2500 | ||
|---|---|---|---|---|
| CAS Number | 112859-71-9 | Molecular Weight | 290.42 | |
| Density | 1.09g/cm3 | Boiling Point | 382.5ºC at 760mmHg | |
| Molecular Formula | C19H27FO | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 207.3ºC | |
Use of HE-2500Fluasterone is a potent G6PD inhibitor with a Ki of 0.51 μM. Fluasterone has anti-inflammatory, cancer preventive, and anti-diabetic effects. Fluasterone is orally active[1][2][3]. |
| Name | Fluasterone |
|---|---|
| Synonym | More Synonyms |
| Description | Fluasterone is a potent G6PD inhibitor with a Ki of 0.51 μM. Fluasterone has anti-inflammatory, cancer preventive, and anti-diabetic effects. Fluasterone is orally active[1][2][3]. |
|---|---|
| Related Catalog | |
| Target |
Ki: 0.51 μM (G6PD)[3] |
| In Vivo | Fluasterone (0.2% and 0.3%; in diet for 39 days) 对糖尿病小鼠有抗高血糖作用[2]。 Fluasterone (200 μg/mouse; intradermal injection; once) 抑制 TPA 诱导的急性炎症和表皮增生作用[3]。 Animal Model: Male C57BL/KsJ db/db mice, diabetic model[2] Dosage: 0.2% and 0.3% Administration: In the diet for 39 days Result: Markedly reduced plasma glucose levels. |
| References |
| Density | 1.09g/cm3 |
|---|---|
| Boiling Point | 382.5ºC at 760mmHg |
| Molecular Formula | C19H27FO |
| Molecular Weight | 290.42 |
| Flash Point | 207.3ºC |
| Exact Mass | 290.20500 |
| PSA | 17.07000 |
| LogP | 4.85640 |
| Vapour Pressure | 4.7E-06mmHg at 25°C |
| Index of Refraction | 1.529 |
| 16-fluoro-5-androsten-17-one |