CGP 20712 dihydrochloride

Modify Date: 2024-03-09 12:33:31

CGP 20712 dihydrochloride Structure
CGP 20712 dihydrochloride structure
Common Name CGP 20712 dihydrochloride
CAS Number 1216905-73-5 Molecular Weight 567.39
Density N/A Boiling Point N/A
Molecular Formula C23H27Cl2F3N4O5 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CGP 20712 dihydrochloride


CGP 20712 dihydrochloride is an antagonist of β 3-adrenoceptor. CGP 20712 dihydrochloride inhibits isoproterenol with the IC50 of 79 μM[1].

 Names

Name 2-Hydroxy-5-{2-[(2-hydroxy-3-{4-[1-methyl-4-(trifluoromethyl)-1H-imidazol-2-yl]phenoxy}propyl)amino]ethoxy}benzamide dihydrochloride
Synonym More Synonyms

 CGP 20712 dihydrochloride Biological Activity

Description CGP 20712 dihydrochloride is an antagonist of β 3-adrenoceptor. CGP 20712 dihydrochloride inhibits isoproterenol with the IC50 of 79 μM[1].
Related Catalog
References

[1]. Van Liefde I, et al. Isoproterenol and selective agonists stimulate similar atypical beta-adrenoceptors in rat adipocytes. Biochem Pharmacol. 1993 Feb 24;45(4):974-7.  

 Chemical & Physical Properties

Molecular Formula C23H27Cl2F3N4O5
Molecular Weight 567.39
Exact Mass 566.131042

 Synonyms

Benzamide, 2-hydroxy-5-[2-[[2-hydroxy-3-[4-[1-methyl-4-(trifluoromethyl)-1H-imidazol-2-yl]phenoxy]propyl]amino]ethoxy]-, hydrochloride (1:2)
2-Hydroxy-5-{2-[(2-hydroxy-3-{4-[1-methyl-4-(trifluoromethyl)-1H-imidazol-2-yl]phenoxy}propyl)amino]ethoxy}benzamide dihydrochloride