CKD-519

Modify Date: 2024-01-10 09:19:40

CKD-519 Structure
CKD-519 structure
Common Name CKD-519
CAS Number 1402796-27-3 Molecular Weight 601.60
Density N/A Boiling Point N/A
Molecular Formula C31H34F7NO3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of CKD-519


CKD-519 is a selective and potent cholesteryl ester transfer protein (CETP) inhibitor, which inhibits CETP-mediated transfer of cholesteryl ester in human serum with an IC50 of 2.3 nM[1].

 Names

Name CKD-519

 CKD-519 Biological Activity

Description CKD-519 is a selective and potent cholesteryl ester transfer protein (CETP) inhibitor, which inhibits CETP-mediated transfer of cholesteryl ester in human serum with an IC50 of 2.3 nM[1].
Related Catalog
Target

IC50: 2.3 nM (Cholesteryl ester transfer protein)[1]

References

[1]. Kim CO, et al. Pharmacokinetics, pharmacodynamics and safety of CKD-519, a CETP inhibitor, in healthy subjects. Drug Des Devel Ther. 2016 Nov 15;10:3763-3770.

 Chemical & Physical Properties

Molecular Formula C31H34F7NO3
Molecular Weight 601.60