MCT1-IN-4a

Modify Date: 2024-04-07 17:57:17

MCT1-IN-4a Structure
MCT1-IN-4a structure
Common Name MCT1-IN-4a
CAS Number 1448314-00-8 Molecular Weight 385.419
Density N/A Boiling Point N/A
Molecular Formula C24H19NO4 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of MCT1-IN-4a


MCT1-IN-4a is a potent, selective monocarboxylate transporter 1 (MCT1) inhibitor with IC50 of 90 nM; exhibits significant single agent activity in MCT1 expressing GL261-luc2 syngraft model, but not in MCT4 expressing MDA-MB-231 xenograft model; has good absorption, metabolic stability, and a low drug efflux ratio.

 Names

Name MCT1-IN-4a

 MCT1-IN-4a Biological Activity

Description MCT1-IN-4a is a potent, selective monocarboxylate transporter 1 (MCT1) inhibitor with IC50 of 90 nM; exhibits significant single agent activity in MCT1 expressing GL261-luc2 syngraft model, but not in MCT4 expressing MDA-MB-231 xenograft model; has good absorption, metabolic stability, and a low drug efflux ratio.
References References 1. Gurrapu S, et al. Bioorg Med Chem Lett. 2016 Jul 15;26(14):3282-6. View Related Products by Target Monocarboxylate Transporter (MCT)

 Chemical & Physical Properties

Molecular Formula C24H19NO4
Molecular Weight 385.419
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