![]() CCR2 antagonist 1 structure
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Common Name | CCR2 antagonist 1 | ||
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CAS Number | 1683534-96-4 | Molecular Weight | 549.47 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C28H32BrF3N2O | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of CCR2 antagonist 1CCR2 antagonist 1 is a high-affinity and long-residence-time CCR2 antagonist, with a Ki of 2.4 nM. |
Name | CCR2 antagonist 1 |
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Description | CCR2 antagonist 1 is a high-affinity and long-residence-time CCR2 antagonist, with a Ki of 2.4 nM. |
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Related Catalog | |
Target |
CCR2:2.4 nM (Ki) |
In Vitro | The combination of SAR and SKR in the hit-to-lead process results in the discovery of a new higheaffinity and longeresidenceetime CCR2 antagonist (CCR2 antagonist 1 (compound 15a), Ki=2.4 nM; RT=714 min)[1]. |
References |
Molecular Formula | C28H32BrF3N2O |
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Molecular Weight | 549.47 |