PROTAC BET degrader-2
Modify Date: 2024-01-13 09:55:37
PROTAC BET degrader-2 structure
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Common Name | PROTAC BET degrader-2 | ||
|---|---|---|---|---|
| CAS Number | 2093388-33-9 | Molecular Weight | 770.84 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C41H42N10O6 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PROTAC BET degrader-2PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins with an IC50 value of 9.6 nM in cell growth inhibition in the RS4;11 cells and capable of achieving tumor regression. |
| Name | PROTAC BET degrader-2 |
|---|
| Description | PROTAC BET degrader-2 is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins with an IC50 value of 9.6 nM in cell growth inhibition in the RS4;11 cells and capable of achieving tumor regression. |
|---|---|
| Related Catalog | |
| Target |
IC50: 9.6 nM (BET in the RS4;11 leukemia cell line)[1]. |
| In Vitro | PROTAC BET degrader-2 (compound 25) is a highly potent degrader of Bromodomain and Extra-Terminal (BET) proteins with an IC50 value of 9.6 nM in cell growth inhibition in the RS4;11 cells and capable of achieving tumor regression[1]. |
| References |
| Molecular Formula | C41H42N10O6 |
|---|---|
| Molecular Weight | 770.84 |
| Storage condition | 2-8℃ |