LSD1-IN-11p structure
|
Common Name | LSD1-IN-11p | ||
|---|---|---|---|---|
| CAS Number | 2101951-67-9 | Molecular Weight | 420.473 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C22H24N6O3 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of LSD1-IN-11pLSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%). |
| Name | LSD1-IN-11p |
|---|
| Description | LSD1-IN-11p is a reversible LSD1 inhibitor with IC50/Kd of 79/21 nM; upregulates the expression of the surrogate cellular biomarker CD86 (IC50=0.52 uM); has moderate oral bioavailability in mice (F%=38%). |
|---|---|
| References | References 1. Mould DP, et al. Bioorg Med Chem Lett. 2017 Jul 15;27(14):3190-3195. View Related Products by Target Histone Demethylase |
| Molecular Formula | C22H24N6O3 |
|---|---|
| Molecular Weight | 420.473 |