Epitinib succinate

Modify Date: 2025-08-27 13:58:09

Epitinib succinate structure	Common Name	Epitinib succinate
	CAS Number	2252334-12-4	Molecular Weight	548.59
	Density	N/A	Boiling Point	N/A
	Molecular Formula	C₂₈H₃₂N₆O₆	Melting Point	N/A
	MSDS	N/A	Flash Point	N/A

Use of Epitinib succinate

Epitinib succinate is an orally active and selective epidermal growth factor receptor tyrosine kinase inhibitor (EGFR-TKI) designed for optimal brain penetration. Epitinib succinate can be used for the research of cancer[1][2].

Name	Epitinib succinate

Description	Epitinib succinate is an orally active and selective epidermal growth factor receptor tyrosine kinase inhibitor (EGFR-TKI) designed for optimal brain penetration. Epitinib succinate can be used for the research of cancer[1][2].
Related Catalog	Research Areas >> Cancer Signaling Pathways >> JAK/STAT Signaling >> EGFR Signaling Pathways >> Protein Tyrosine Kinase/RTK >> EGFR
Target	EGFR[2]
In Vitro	Epitinib succinate is an orally active and selective epidermal growth factor receptor tyrosine kinase inhibitor (EGFR-TKI) designed for optimal brain penetration[1][2].
References	[1]. Zhou et al. The safety profile of a selective EGFR TKI epitinib (HMPL-813) in patients with advanced solid tumors and preliminary clinical efficacy in EGFRm+ NSCLC patients with brain metastasis. Journal of Clinical Oncology 2016 34:15_suppl, e20502-e20502 [2]. Zhou et al. Phase I study of the safety and pharmacokinetics of epitinib, an oral EGFR tyrosine kinase inhibitor, in patients with advanced solid tumors. Journal of Clinical Oncology 2013 31:15_suppl, e19042-e19042

Molecular Formula	C₂₈H₃₂N₆O₆
Molecular Weight	548.59
InChIKey	HISXHQFAOANCJX-UHFFFAOYSA-N
SMILES	C#Cc1cccc(Nc2ncnc3cc(OC)c(NC(=O)N4CCN(CC)CC4)cc23)c1.O=C(O)CCC(=O)O

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Shanghai Nianxing Industrial Co., Ltd
China
Product Name: Epitinib succinate
Price: Check
Purity: 98.0%
Delivery: 10 Day
Contact: Yang
Email: sales@echemcloud.com

DC Chemicals Limited
China
Product Name: Epitinib succinate
Price: ￥Inquiry/1g
Purity: 98.9%
Delivery: 1 Day
Contact: Tony Cao
Email: sales@dcchemicals.com

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Price: ￥3500/5 mg

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Epitinib succinate

Use of Epitinib succinate

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Epitinib succinate Biological Activity

Chemical & Physical Properties

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