ERAP2-IN-1
Modify Date: 2024-09-16 22:32:00
ERAP2-IN-1 structure
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Common Name | ERAP2-IN-1 | ||
|---|---|---|---|---|
| CAS Number | 2420551-38-6 | Molecular Weight | 458.45 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C20H21F3N2O5S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of ERAP2-IN-1ERAP2-IN-1 (compound 61) is an uncompetitive ERAP2 inhibitor. ERAP2-IN-1 specifically inhibits the ERAP2 peptide hydrolysis activity, inhibiting Arg-AMC hydrolysis with an IC50 of 27 μM and model peptide hydrolysis with an IC50 of 44 μM[1]. |
| Name | ERAP2-IN-1 |
|---|
| Description | ERAP2-IN-1 (compound 61) is an uncompetitive ERAP2 inhibitor. ERAP2-IN-1 specifically inhibits the ERAP2 peptide hydrolysis activity, inhibiting Arg-AMC hydrolysis with an IC50 of 27 μM and model peptide hydrolysis with an IC50 of 44 μM[1]. |
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| Related Catalog | |
| References |
| Molecular Formula | C20H21F3N2O5S |
|---|---|
| Molecular Weight | 458.45 |
| InChIKey | BGLAMEXMBJAJBI-UHFFFAOYSA-N |
| SMILES | COc1ccc(C(=O)O)cc1S(=O)(=O)Nc1ccc(C(F)(F)F)cc1N1CCCCC1 |