Difelikefalin HCl
Modify Date: 2025-08-25 18:12:17
Difelikefalin HCl structure
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Common Name | Difelikefalin HCl | ||
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| CAS Number | 2711717-77-8 | Molecular Weight | 789.237 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C36H56Cl3N7O6 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Difelikefalin HClDifelikefalin is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM). Difelikefalin is selective for KOR over the μ-opioid receptor. |
| Name | Difelikefalin HCl |
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| Description | Difelikefalin is a κ-opioid receptor (KOR) agonist. It activates KOR in HEK293 cells expressing the human receptor (EC50 = 0.16 nM in a transactivation assay) and inhibits forskolin-induced cAMP production in R1.G1 mouse thyoma cells (EC50 = 0.048 nM). Difelikefalin is selective for KOR over the μ-opioid receptor. |
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| Molecular Formula | C36H56Cl3N7O6 |
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| Molecular Weight | 789.237 |