Histone Acetyltransferase Inhibitor II

Modify Date: 2024-01-13 17:32:59

Histone Acetyltransferase Inhibitor II Structure
Histone Acetyltransferase Inhibitor II structure
Common Name Histone Acetyltransferase Inhibitor II
CAS Number 932749-62-7 Molecular Weight 464.14700
Density N/A Boiling Point N/A
Molecular Formula C20H16Br2O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Histone Acetyltransferase Inhibitor II


Histone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 µM; Histone Acetyltransferase Inhibitor II can be used in cancer research.

 Names

Name 2,6-bis(3-bromo-4-hydroxybenzylidene)cyclohexanone
Synonym More Synonyms

 Histone Acetyltransferase Inhibitor II Biological Activity

Description Histone Acetyltransferase Inhibitor II is a potent and cell permeable p300 inhibitor, with an IC50 of 5 µM; Histone Acetyltransferase Inhibitor II can be used in cancer research.
Related Catalog
Target

IC50:5 µM (p300)[1]

In Vitro Histone Acetyltransferase Inhibitor II 是一种有效的,细胞渗透的 p300 抑制剂,IC50 值为 5 µM,可用于癌症研究。
References

[1]. Costi R, et al. Cinnamoyl compounds as simple molecules that inhibit p300 histone acetyltransferase. J Med Chem. 2007 Apr 19;50(8):1973-7. Epub 2007 Mar 10.

 Chemical & Physical Properties

Molecular Formula C20H16Br2O3
Molecular Weight 464.14700
Exact Mass 461.94700
PSA 57.53000
LogP 5.84280
Storage condition 2-8℃

 Synonyms

HistoneAcetyltransferaseInhibitorII
Histone Acetyltransferase Inhibitor II