PKC-theta inhibitor 1
Modify Date: 2025-08-25 18:58:02
PKC-theta inhibitor 1 structure
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Common Name | PKC-theta inhibitor 1 | ||
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| CAS Number | 1160501-81-4 | Molecular Weight | 348.32 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C17H15F3N4O | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PKC-theta inhibitor 1PKC-theta inhibitor 1 is the PKCθ inhibitor with an Ki value of 6 nM, inhibits IL-2 production in vivo with an IC50 of 0.19 μM. PKC-theta inhibitor 1 demonstrates a reduction of symptoms in a mouse model of multiple sclerosis[1]. |
| Name | PKC-theta inhibitor 1 |
|---|
| Description | PKC-theta inhibitor 1 is the PKCθ inhibitor with an Ki value of 6 nM, inhibits IL-2 production in vivo with an IC50 of 0.19 μM. PKC-theta inhibitor 1 demonstrates a reduction of symptoms in a mouse model of multiple sclerosis[1]. |
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| Related Catalog | |
| Target |
PKCθ:6 nM (Ki) PKCδ:392 μM (Ki) PKCα:1020 μM (Ki) IL-2 production:0.19 μM (IC50) |
| References |
| Molecular Formula | C17H15F3N4O |
|---|---|
| Molecular Weight | 348.32 |