CJ-1639
Modify Date: 2023-10-20 10:34:26
CJ-1639 structure
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Common Name | CJ-1639 | ||
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| CAS Number | 1313759-88-4 | Molecular Weight | 478.655 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C27H34N4O2S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of CJ-1639CJ-1639 (CJ1639) is a potent, highly selective dopamine D3 receptor (D3R) full agonist with Ki of 0.5 nM, >5,000-fold selectivity over D1 and D2 receptors in binding assays.CJ-1639 binds to human D3 receptor with a K(i) value of 3.61 nM and displays over >1000-fold selectivity over human D1 and D2 receptors.CJ-1639 is an excellent pharmacological tool to elucidate the role of the D3 receptor in different neurological conditions in animal models. |
| Name | CJ-1639 |
|---|
| Description | CJ-1639 (CJ1639) is a potent, highly selective dopamine D3 receptor (D3R) full agonist with Ki of 0.5 nM, >5,000-fold selectivity over D1 and D2 receptors in binding assays.CJ-1639 binds to human D3 receptor with a K(i) value of 3.61 nM and displays over >1000-fold selectivity over human D1 and D2 receptors.CJ-1639 is an excellent pharmacological tool to elucidate the role of the D3 receptor in different neurological conditions in animal models. |
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| References | 1. Jianyong Chen, et al. ACS Med Chem Lett. 2011 Aug 11;2(8):620-625. |
| Molecular Formula | C27H34N4O2S |
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| Molecular Weight | 478.655 |