PDE10A-IN-31 structure
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Common Name | PDE10A-IN-31 | ||
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CAS Number | 1639889-98-7 | Molecular Weight | 477.524 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C28H23N5O3 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of PDE10A-IN-31PDE10A-IN-31 is a potent, highly selective PDE10A inhibitor with IC50 of 2 nM for both rPDE10A and hPDE10A; dispalys >2,000-fold selective over PDE1B/2A/3B/4D/5A/7A9A, weak activity on CYP isoforms; displays excellent pharmacokinetic properties. |
Name | PDE10A-IN-31 |
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Description | PDE10A-IN-31 is a potent, highly selective PDE10A inhibitor with IC50 of 2 nM for both rPDE10A and hPDE10A; dispalys >2,000-fold selective over PDE1B/2A/3B/4D/5A/7A9A, weak activity on CYP isoforms; displays excellent pharmacokinetic properties. |
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References | References 1. Meegalla SK, et al. Bioorg Med Chem Lett. 2016 Sep 1;26(17):4216-22. View Related Products by Target Phosphodiesterase (PDE) |
Molecular Formula | C28H23N5O3 |
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Molecular Weight | 477.524 |