Cyclic Arg-Gly-Asp-D-Tyr-Lys structure
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Common Name | Cyclic Arg-Gly-Asp-D-Tyr-Lys | ||
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CAS Number | 250612-42-1 | Molecular Weight | 847.72 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C31H43F6N9O12 | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of Cyclic Arg-Gly-Asp-D-Tyr-LysCyclo(RGDyK) trifluoroacetate is a potent and selective αVβ3 integrin inhibitor with an IC50 of 20 nM. |
Name | Cyclo(RGDyK) |
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Synonym | More Synonyms |
Description | Cyclo(RGDyK) trifluoroacetate is a potent and selective αVβ3 integrin inhibitor with an IC50 of 20 nM. |
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Related Catalog | |
Target |
IC50: 20 nM (αVβ3 Integrin), 3000 nM (αIIbβ3 Integrin), 4000 nM (αVβ5 Integrin)[1] |
In Vitro | Cyclo(RGDyK) (c(RGDyK(SAA)) shows high affinity and selectivity for αVβ3 over αVβ5 (IC50=4000 nM) and αIIbβ3 (IC50=3000 nM)[1]. |
References |
Molecular Formula | C31H43F6N9O12 |
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Molecular Weight | 847.72 |
Storage condition | -20℃ |
Cyclic Arg-Gly-Asp-D-Tyr-Lys |