PBRM1-BD2-IN-4

Modify Date: 2024-04-05 17:16:11

PBRM1-BD2-IN-4 Structure
PBRM1-BD2-IN-4 structure
Common Name PBRM1-BD2-IN-4
CAS Number 2819989-60-9 Molecular Weight 272.73
Density N/A Boiling Point N/A
Molecular Formula C15H13ClN2O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of PBRM1-BD2-IN-4


PBRM1-BD2-IN-4 (compound 15) is a potent PBRM1 Bromodomain inhibitor with Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.2 μM for PBRM1-BD2. PBRM1-BD2-IN-4 can be used to research anticancer[1].

 Names

Name PBRM1-BD2-IN-4

 PBRM1-BD2-IN-4 Biological Activity

Description PBRM1-BD2-IN-4 (compound 15) is a potent PBRM1 Bromodomain inhibitor with Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.2 μM for PBRM1-BD2. PBRM1-BD2-IN-4 can be used to research anticancer[1].
Related Catalog
Target

Kd: 5.5 μM (PBRM1-BD2), 11.1 μM (PBRM1-BD5)[1] IC50: 0.2 μM (PBRM1-BD2)[1]

 Chemical & Physical Properties

Molecular Formula C15H13ClN2O
Molecular Weight 272.73