PBRM1-BD2-IN-4 structure
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Common Name | PBRM1-BD2-IN-4 | ||
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CAS Number | 2819989-60-9 | Molecular Weight | 272.73 | |
Density | N/A | Boiling Point | N/A | |
Molecular Formula | C15H13ClN2O | Melting Point | N/A | |
MSDS | N/A | Flash Point | N/A |
Use of PBRM1-BD2-IN-4PBRM1-BD2-IN-4 (compound 15) is a potent PBRM1 Bromodomain inhibitor with Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.2 μM for PBRM1-BD2. PBRM1-BD2-IN-4 can be used to research anticancer[1]. |
Name | PBRM1-BD2-IN-4 |
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Description | PBRM1-BD2-IN-4 (compound 15) is a potent PBRM1 Bromodomain inhibitor with Kd values of 5.5 μM and 11.1 μM for PBRM1-BD2 and PBRM1-BD5, respectively, and an IC50 value of 0.2 μM for PBRM1-BD2. PBRM1-BD2-IN-4 can be used to research anticancer[1]. |
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Related Catalog | |
Target |
Kd: 5.5 μM (PBRM1-BD2), 11.1 μM (PBRM1-BD5)[1] IC50: 0.2 μM (PBRM1-BD2)[1] |
Molecular Formula | C15H13ClN2O |
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Molecular Weight | 272.73 |