Ac-RYYRWK-NH2 TFA
Modify Date: 2024-01-02 12:12:22
Ac-RYYRWK-NH2 TFA structure
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Common Name | Ac-RYYRWK-NH2 TFA | ||
|---|---|---|---|---|
| CAS Number | 408305-09-9 | Molecular Weight | 1126.19 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C51H70F3N15O11 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of Ac-RYYRWK-NH2 TFAAc-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for µ-, κ- or δ-opioid receptors[1]. |
| Name | Ac-RYYRWK-NH2 TFA |
|---|
| Description | Ac-RYYRWK-NH2 is a potent and selective partial agonist for the nociceptin receptor (NOP), [3H]Ac-RYYRWK-NH2 binds to rat cortical membranes ORL1 with a Kd of 0.071 nM, but has no affinity for µ-, κ- or δ-opioid receptors[1]. |
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| Related Catalog | |
| In Vitro | [3H]ac-RYYRWK-NH2 binding to rat cortical membranes revealed a single high affinity site for [3H]ac-RYYRWK-NH2 (Kd=0.071 nM)[1]. Naloxone benzoylhydrazone displaced [3H]acRYYRWK-NH2 binding to rat cortical membranes (Ki=104 nM) and human ORL1 (Ki=136 nM) as well as [125I]Tyr14-NC-OH to ORL1 (Ki=37 nM) has no affinity for µ-, κ- or δ-opioid receptors[1]. |
| References |
| Molecular Formula | C51H70F3N15O11 |
|---|---|
| Molecular Weight | 1126.19 |