PCAF-IN-2
Modify Date: 2024-01-02 20:31:42
PCAF-IN-2 structure
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Common Name | PCAF-IN-2 | ||
|---|---|---|---|---|
| CAS Number | 56173-05-8 | Molecular Weight | 268.20 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C10H7F3N6 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of PCAF-IN-2PCAF-IN-2 (compound 17) is a potent PCAF inhibitor with an IC50 value of 5.31 µM. PCAF-IN-2 shows anti-tumour activity. CAF-IN-2 induces apoptosis and arrest the cell cycle at the G2/M phase[1]. |
| Name | PCAF-IN-2 |
|---|
| Description | PCAF-IN-2 (compound 17) is a potent PCAF inhibitor with an IC50 value of 5.31 µM. PCAF-IN-2 shows anti-tumour activity. CAF-IN-2 induces apoptosis and arrest the cell cycle at the G2/M phase[1]. |
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| Related Catalog | |
| Target |
PCAF:5.31 μM (IC50) |
| In Vitro | PCAF-IN-2 shows anti-tumour activity with IC50s of 3.06, 5.69, 7.56, 2.83 µM for HePG2, MCF-7, PC3, HCT-116 cells, respectively[1]. PCAF-IN-2 (10 µM; 24 h) induces apoptosis and arrest the cell cycle at the G2/M phase in HePG2 cells[1]. |
| References |
| Molecular Formula | C10H7F3N6 |
|---|---|
| Molecular Weight | 268.20 |