GSK 2250665A
Modify Date: 2025-09-03 19:48:30
GSK 2250665A structure
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Common Name | GSK 2250665A | ||
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| CAS Number | 1246030-96-5 | Molecular Weight | 459.606 | |
| Density | 1.3±0.1 g/cm3 | Boiling Point | 676.6±65.0 °C at 760 mmHg | |
| Molecular Formula | C26H29N5OS | Melting Point | N/A | |
| MSDS | N/A | Flash Point | 363.0±34.3 °C | |
Use of GSK 2250665AGSK-2250665A (Compound 13) is a selective Itk inhibitor with a pKi of 9.2. |
| Name | trans-4-({4-Benzyl-6-[(6-ethyl-1,3-benzothiazol-2-yl)amino]-2-pyrimidinyl}amino)cyclohexanol |
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| Synonym | More Synonyms |
| Description | GSK-2250665A (Compound 13) is a selective Itk inhibitor with a pKi of 9.2. |
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| Related Catalog | |
| In Vitro | GSK-2250665A (Compound 13) achieves a pIC50 of 7.3 in the cell assay, measuring inhibition of IFNγ production from PBMCs (Peripheral Blood Mononuclear Cells) [1]. |
| References |
| Density | 1.3±0.1 g/cm3 |
|---|---|
| Boiling Point | 676.6±65.0 °C at 760 mmHg |
| Molecular Formula | C26H29N5OS |
| Molecular Weight | 459.606 |
| Flash Point | 363.0±34.3 °C |
| Exact Mass | 459.209290 |
| LogP | 5.31 |
| Vapour Pressure | 0.0±2.2 mmHg at 25°C |
| Index of Refraction | 1.713 |
| trans-4-({4-Benzyl-6-[(6-ethyl-1,3-benzothiazol-2-yl)amino]-2-pyrimidinyl}amino)cyclohexanol |
| Cyclohexanol, 4-[[4-[(6-ethyl-2-benzothiazolyl)amino]-6-(phenylmethyl)-2-pyrimidinyl]amino]-, trans- |