Keap1-Nrf2-IN-3

Modify Date: 2024-01-10 20:09:06

Keap1-Nrf2-IN-3 Structure
Keap1-Nrf2-IN-3 structure
Common Name Keap1-Nrf2-IN-3
CAS Number 2095066-47-8 Molecular Weight 538.64
Density N/A Boiling Point N/A
Molecular Formula C31H34N6O3 Melting Point N/A
MSDS N/A Flash Point N/A

 Use of Keap1-Nrf2-IN-3


Keap1-Nrf2-IN-3 is a KEAP1:NRF2 protein−protein interaction inhibitor, and with a Kd value of 2.5 nM for KEAP1 protein.

 Names

Name Keap1-Nrf2-IN-3

 Keap1-Nrf2-IN-3 Biological Activity

Description Keap1-Nrf2-IN-3 is a KEAP1:NRF2 protein−protein interaction inhibitor, and with a Kd value of 2.5 nM for KEAP1 protein.
Related Catalog
References

[1]. Norton D, et al. Fragment-Guided Discovery of Pyrazole Carboxylic Acid Inhibitors of the Kelch-like ECH-Associated Protein 1: Nuclear Factor Erythroid 2 Related Factor 2 (KEAP1:NRF2) Protein-Protein Interaction. J Med Chem. 2021 Nov 11;64(21):15949-15972.

 Chemical & Physical Properties

Molecular Formula C31H34N6O3
Molecular Weight 538.64