RSK2-IN-2

Modify Date: 2024-09-23 20:44:51

RSK2-IN-2 Structure
RSK2-IN-2 structure
 Common Name RSK2-IN-2
CAS Number 1637749-78-0 Molecular Weight 289.29
Density N/A Boiling Point N/A
Molecular Formula C16H11N5O Melting Point N/A
MSDS N/A Flash Point N/A

 Use of RSK2-IN-2


RSK2-IN-2 (Compound 25) is a reversible covalent inhibitor of the RPS6KA3 (RSK2) kinase. RSK2-IN-2 is also described to inhibit MSK1, MSK2 and RSK3[1].

 Names

Name RSK2-IN-2

 RSK2-IN-2 Biological Activity

Description RSK2-IN-2 (Compound 25) is a reversible covalent inhibitor of the RPS6KA3 (RSK2) kinase. RSK2-IN-2 is also described to inhibit MSK1, MSK2 and RSK3[1].
Related Catalog
Target

RSK2

RSK3

MSK1

MSK2

In Vitro RSK2-IN-2 (Compound 25) shows strong activity with ERK2-MSK1 cascade pIC50 of 9.6[1].
References

[1]. Hall A, et al. Discovery and Characterization of a Novel Series of Chloropyrimidines as Covalent Inhibitors of the Kinase MSK1. ACS Med Chem Lett. 2022 Jun 25;13(7):1099-1108.

 Chemical & Physical Properties

Molecular Formula C16H11N5O
Molecular Weight 289.29
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Chemsrc provides RSK2-IN-2(CAS#:1637749-78-0) MSDS, density, melting point, boiling point, structure, formula, molecular weight etc. Articles of RSK2-IN-2 are included as well.>> amp version: RSK2-IN-2

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