IACS-9571
Modify Date: 2024-01-02 06:37:40
IACS-9571 structure
|
Common Name | IACS-9571 | ||
|---|---|---|---|---|
| CAS Number | 1800477-30-8 | Molecular Weight | 642.76 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C32H42N4O8S | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of IACS-9571IACS-9571 is a potent and selective inhibitor of TRIM24 and BRPF1, with IC50 of 8 nM for TRIM24, and Kds of 31 nM and 14 nM for TRIM24 and BRPF1, respectively. |
| Name | IACS-9571 |
|---|
| Description | IACS-9571 is a potent and selective inhibitor of TRIM24 and BRPF1, with IC50 of 8 nM for TRIM24, and Kds of 31 nM and 14 nM for TRIM24 and BRPF1, respectively. |
|---|---|
| Related Catalog | |
| Target |
IC50: 8 nM (TRIM24)[1] Kd: 31 nM (TRIM24), 14 nM (BRPF1)[1] |
| In Vitro | IACS-9571 shows excellent cellular potency with EC50 of 50 nM. IACS-9571 (1 μM) has potent activities against a panel of 32 bromodomains. IACS-9571 is a selective dual TRIM24/BRPF1 inhibitor (Kd = 1.3/2.1 nM) with 9- and 21-fold selectivity against BRPF2 and BRPF3, respectively. IACS-9571 does not interact with the BET sub-family of bromodomains, displaying greater than 7,700-fold selectivity versus BRD4(1, 2) relative to TRIM24[1]. |
| References |
| Molecular Formula | C32H42N4O8S |
|---|---|
| Molecular Weight | 642.76 |
| Storage condition | 2-8℃ |
- Shanghai Nianxing Industrial Co., Ltd
- China
- Product Name: IACS-9571
- Price: Negotiable
- Purity: 98.0%
- Delivery: 10 Day
- Contact: Huang
- Email: sales@echemcloud.com
- ShangHai DC Chemicals Co.,Ltd
- China
- Product Name: IACS-9571
- Price: ￥Inquiry/1g
- Purity: 98.9%
- Delivery: 1 Day
- Contact: Tony Lai
- Email: order@dcchemicals.com
- DC Chemicals Limited
- China
- Product Name: IACS-9571
- Price: $Inquiry/100mg $Inquiry/250mg $Inquiry/500mg
- Purity: 98.0%
- Delivery: 3 Day
- Contact: Tony Cao
- Email: sales@dcchemicals.com
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Price: $180/1mg
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