APJ receptor agonist 6
Modify Date: 2024-08-14 17:50:16
APJ receptor agonist 6 structure
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Common Name | APJ receptor agonist 6 | ||
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| CAS Number | 1965244-85-2 | Molecular Weight | 523.60 | |
| Density | N/A | Boiling Point | N/A | |
| Molecular Formula | C29H34FN3O5 | Melting Point | N/A | |
| MSDS | N/A | Flash Point | N/A | |
Use of APJ receptor agonist 6APJ receptor agonist 6 (compound 9) is a potent APJ (apelin receptor) agonist, with Ki of 1.3 μM. APJ receptor agonist 6 has EC50 values of 0.070 , 0.097, and 0.063 μM for calcium, cAMP, and β-arrestin, respectively[1]. |
| Name | APJ receptor agonist 6 |
|---|
| Description | APJ receptor agonist 6 (compound 9) is a potent APJ (apelin receptor) agonist, with Ki of 1.3 μM. APJ receptor agonist 6 has EC50 values of 0.070 , 0.097, and 0.063 μM for calcium, cAMP, and β-arrestin, respectively[1]. |
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| Related Catalog | |
| Target |
EC50: 0.800 ± 0.1 μM (Apelin Receptor calcium), 0.844 ± 0.2 μM (Apelin Receptor cAMP), 6.22 ± 2.0 μM (Apelin Receptor β-arrestin), >10 μM (AT1 calcium)[1] |
| References |
| Molecular Formula | C29H34FN3O5 |
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| Molecular Weight | 523.60 |